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GLP-1 · APPROVED

Liraglutide

ALSO KNOWN AS · Victoza · Saxenda

The first-generation once-daily GLP-1 agonist, now largely superseded by weekly agents but still widely used and available as a generic in several markets.

Mechanism

Liraglutide is 97% homologous to native GLP-1 with a C16 palmitoyl chain that supports albumin binding and self-association at the injection site, extending exposure to roughly a day.

Clinical evidence

SCALE reported a mean 8.0% weight reduction at 56 weeks on 3.0 mg. LEADER demonstrated a reduction in cardiovascular death in type 2 diabetes, the first such result for the class.

PRIMARY SOURCES

  1. 01SCALE obesity trialNew England Journal of Medicine
  2. 02LEADER trialNew England Journal of Medicine

Educational reference only. Trial figures are protocol-condition means, not individual predictions. Investigational compounds are not approved medicines and have no legitimate consumer supply route.